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Saw Palmetto × Beta-2 Agonists

MODERATE INTERACTION

⚠️ Mechanism

Saw Palmetto is a weak inhibitor of CYP3A4, which decreases metabolism of CYP3A4 substrates, potentially increasing their plasma concentrations and risk of adverse effects.

📋 Effect

Increased plasma levels of salmeterol (beta2-agonists), potentially leading to toxicity or enhanced adverse effects.

💊 Management

Monitor for increased adverse effects of salmeterol. Dose reduction may be necessary. Consider alternative supplement or consult healthcare provider.

Plain Language Summary

This combination carries a moderate risk of increasing the side effects of your medication. Saw Palmetto can slow down how your body breaks down beta-2 agonists, which may lead to higher levels of the drug in your bloodstream.

Source

Flockhart CYP450 Table (drug-interactions.medicine.iu.edu)

Supporting Research

Serenoa repens for benign prostatic hyperplasia PMID:19370565 DOI:10.1002/14651858.CD001423.pub2 2009
Serenoa repens for benign prostatic hyperplasia PMID:23235581 DOI:10.1002/14651858.CD001423.pub3 2012
Non-hormonal treatment for male infertility: the potential role of Serenoa repens, selenium and lycopene PMID:31002161 DOI:10.26355/eurrev_201904_17595 2019
Comparison of Serenoa repens With Tamsulosin in the Treatment of Benign Prostatic Hyperplasia: A Systematic Review and Meta-Analysis PMID:32274957 DOI:10.1177/1557988320905407 2020
Effects of dietary supplements on androgenetic alopecia: a systematic review and network meta-analysis PMID:41561175 DOI:10.3389/fnut.2025.1719711 2025
Benign prostate hyperplasia and nutrition PMID:31451276 DOI:10.1016/j.clnesp.2019.07.015 2019
American palm ethnomedicine: a meta-analysis PMID:20034398 DOI:10.1186/1746-4269-5-43 2009
Benign prostatic hyperplasia and male lower urinary tract symptoms (LUTS) PMID:21871136 2011
Medical Disclaimer: This interaction record is for informational and educational purposes only and does not constitute medical advice. Drug-supplement interactions can be dangerous. Always consult your healthcare provider or pharmacist before combining any supplement with prescription medications. Do not stop or change any medication without professional guidance.